Sl. No. | Intermediate Name | Product Name | CAS Number |
---|---|---|---|
1 | 2-chloromethyl-3-methyl-4- (2,2,2-trifluoroethoxy) pyridine hydrochloride(Lansoprazole chloro compound) | Lansoprazole | 127337-60-4 |
2 | 2-[[[3-methyl-4-(2,2,2-trifluoroethoxy) pyridine-2-yl] methyl]thio]-1H-benzimidazole (Lansoprazole Sulphide compound) | Lansoprazole | 103577-40-8 |
3 | 2-(Chloromethyl)-3,4-dimethoxy pyridine hydrochloride(Pantoprazole Chloro Compound) | Pantoprazole sodium | 72830-09-2 |
4 | 5-(difluoromethoxy)-2-[[[3,4-dimethoxy-2-pyridinyl]methyl] thio]-1H-benzimidazole (Pantoprazole Sulphide compound) | Pantoprazole sodium | 102625-64-9 |
5 | 2-[[[4-(3-methoxypropoxy)-3-methyl-2-pyridinyl] methyl] thio]-1H-benzimidazole (Rabeprazole Sulphide compound) | Rabeprazole | 117977-21-6 |
6 | Cis-[2-(2,4-dichlorophenyl)-2-(1H-1,2,4-triazol-1-yl-methyl)-1,3-dioxolan -4-yl] methanol-p-Toluenesulfonate | Terconazole Itraconazole |
103661-14-9 |
7 | 4-(4-Hydroxy phenyl)-1-(1-methylethyl)piperazine | Terconazole | 67914-97-0 |
8 | (R*,S*)-2-(2,4-difluorophenyl)-3-(5-fluoropyrimidine-4-yl)-1-(1H-1,2,4-triazol-1-yl) butan-2-ol | Voriconazole | 188416-29-7 |
9 | 2-(2,4-difluorophenyl)-3-(4-chloro-5-fluoro pyrimidine-4-yl)-1-(1H-1,2,4-triazol-1-yl) butan-2-ol hydrochloride | Voriconazole | 188416-35-5 |
10 | (S)-3-(dimethylamino)-1-(thiophen-2-yl) propan-1-ol-2-hydroxy-2-phenylacetate | Duloxetine Hydrochloride | 287737-72-8 |
11 | 2-(2-Nitro anilino)-5-methyl thiophene-3-carbonitrile | Olanzapine | 138564-59-7 |
12 | 4-amino-2-methyl-10H-thieno [2,3-b] [1,5] benzodiazepine hydrochloride | Olanzapine | 138564-60-0 |
13 | 7-(4-bromo butoxy)-3,4-dihydro carbostyril | Aripiprazole | 29722-34-5 |
14 | (R)-5-(2-aminopropyl)-2-methoxy-benzenesulfonamide | Tamsulosin HCl | 112101-81-2 |
15 | 1-(2-bromoethoxy)-2-ethoxy-benzene | Tamsulosin HCl | 3259-03-8 |
16 | (R)-5-bromo-3-[(1-methyl-2-pyrrolidinyl)methyl]-1H-indole | Eletriptan | 143322-57-0 |
17 | 2-Bromo-1-cyclopropyl-2-(2-fluorophenyl)ethanone | Prasugrel | 204205-33-4 |
18 | Benzoic acid, 3-[(1R)-3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-(phenylmethoxy)-, methyl ester | Fesoterodine Fumerate | 156755-35-0 |
19 | (+)-N,N-Diisopropyl-3-(2-hydroxy-5-hydroxymethylphenyl)-3-phenylpropylamine | Fesoterodine Fumerate | 207679-81-0 |
20 | N-[3-amino-4-(methylamino)benzoyl]-N-2-pyridinyl-, ethyl ester | Dabigatran | 212322-56-0 |
21 | 2-(n-Butyl)-3-(4-hydroxybenzoyl)-5-nitrobenzofuran | Dronedarone | 141645-16-1 |
22 | Methyl 2-[1-[[(benzyloxy)carbonyl]amino]-1-methylethyl]-5,6-dihydroxypyrimidine-4-carboxylate | Raltegravir | 519032-08-7 |
23 | Methyl 2-[1-[[(benzyloxy)carbonyl]amino]-1-methylethyl]-1-Methyl-5-Hydroxy-6-Oxo-1,6-dihydroxypyrimidine-4-carboxylate | Raltegravir | 888504-27-6 |
24 | Benzyl [1-[4-[[(4-Fluorobenzyl]amino]carbonyl]-5-Hydroxy-1-Methyl-6-Oxo-1,6-Dihydropyrimidine-2-yl]-1-Methylethyl]Carbamate | Raltegravir | 518048-02-7 |
25 | 5-Methyl-1,3,4-Oxadiazole-2-Carboxylic Acid Potassium Salt | Raltegravir | 888504-28-7 |
26 | (1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester | Saxagliptan | 361440-67-7 |
27 | (1S,3S,5S)-2-Azabicyclo[3.1.0]hexane-3-carboxamide | Saxagliptan | 361440-68-8 |
28 | (1S,3S,5S)-2-Azabicyclo[3.1.0]hexane-3-carboxamide, 2,2,2-trifluoroacetate (1:1) | Saxagliptan | 361440-69-9 |
29 | (aS)-a-[[(1,1-dimethylethoxy)carbonyl]amino]-3-hydroxytricyclo[3.3.1.13,7]decane-1-acetic acid | Saxagliptan | 361442-00-4 |
30 | 3-(1-Piperazinyl)-1,2-Benzisothiazole | Lurasidone | 87691-87-0 |
31 | (3aR,4S,7R,7aS) 4,7-Methano-1H-isoindole-1,3(2H)-dione | Lurasidone | 14805-29-9 |
32 | (R,R) Cyclohexane Dicarboxylic Acid | Lurasidone | 46022-05-3 |
33 | (3aR, 7aR)-Hexahydroisobenzofuran-1,3-Dione | Lurasidone | 71749-03-6 |
34 | 2,3,4,5-Tetrahydro-3-(Trifluoroacetyl)-1,5-Methano-1H-3-Benzazepine | Varenicline | 230615-51-7 |
35 | 2,3,4,5-Tetrahydro-1,5-Methano-1H-3-Benzazepine Hydrochloride | Varenicline | 230615-52-8 |
36 | 8-Bromo-7-(But-2-ynyl)-3-Methyl-1H-Purine-2,6(3H,7H)-Dione, | Linagliptin | 666816-98-4 |
37 | 3-(R)-Piperdinyl Pthalimide Hydrochloride | Linagliptin | 886588-61-0 |
38 | (R)-Tert-Butyl piperdin-3-yl Carbamate | Linagliptin | 309956-78-3 |
39 | 1-(Isobutyloxy)ethyl-4-Nitrophenyl Carbonate | Gabapentin | NA |
40 | (1R,2S,5S)-6,6-Dimethyl-3-Aza-Bicyclo[3.1.0]Hexane-2-Carboxylic Acid Methyl Ester Hydrochloride | Boceprevir | 565456-77-1 |
41 | Beta-Amino-Alpha-Hydroxycyclobutanebutanamide Hydrochloride | Boceprevir | 394735-23-0 |
42 | N-[(1,1-dimethylethoxy)carbonyl]-3-methyl-L-valine | Boceprevir | 62965-35-9 |
43 | 1-[N-(2,6-Dimethylphenyl)carbomylmethyl]piperazine | Ranolazine | 5294-61-1 |
44 | (2-methoxyphenoxy)-2,3-Epoxypropane | Ranolazine | 2210-74-4 |
45 | 3-(4-chlorobutyl)-1H-indole-5-carbonitrile | Vilazodone | 143612-79-7 |
46 | Ethyl 5-(piperazin-1-yl)-1-benzofuran-2-carboxylate | Vilazodone | 163521-20-8 |
47 | 4-Oxo-1,4-Dihydroquinoline-3-Carboxylic Acid | Ivacaftor | 13721-01-2 |
48 | 5-Amino-2,4-Di-Tert-Butylphenyl methyl carbonate | Ivacaftor | 1182822-31-6 |
49 | 2-Chloromalonaldehyde | Etoricoxib | 36437-19-1 |
50 | 1-(6-methyl-3-pyridinyl)-2-[4-(methylsulfonyl)phenyl] Ethanone | Etoricoxib | 221615-75-4 |
51 | 4-amino-1- ((2R,3R,4R,5R)-3- fluoro-4-hydroxy-5- (hydroxymethyl)-3-methyltetrahydrofuran- 2-yl)pyrimidin-2(1H)-one | Sofusbuvir | 817204-33-4 |
52 | 1-( 4- iodophenyl ) – piperidine -2- one | Apixaban | 385425-15-0 |
53 | Chloro ( 4- methoxyphenyl ) hydrazono ) acetic acid ethyl ester | Apixaban | 27143-07-3 |
54 | 2-Piperiodone | Apixaban | 675-20-7 |
55 | (S,S)-2,8-Diazabicyclo[4,3,0] nonane | Moxifloxacin Hydrochloride | 151213-40-0 |
56 | 1-cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid ethyl ester | Moxifloxacin Hydrochloride | 112811-71-9 |
57 | (2-[2-[3(S)-[3-[(1E)-2-(7-chloroqunolin-2-yl)phenyl]-3-hydroxypropyl]phenyl-2-propanol) | Montelukast sodium | 142569-70-8 |
58 | (1-(Mercaptomethyl) cyclopropane acetic acid) | Montelukast sodium | 162515-68-6 |